Technical Articles
Biotinylated CRBN/DDB1
What Is Biotinylated CRBN/DDB1: How the Labeled Complex Serves PROTAC Degradation Research
Biotinylated CRBN/DDB1 is the substrate-recognition module of CRL4 E3 ligase, immobilized for binding assays. This article explains its role in PROTAC and molecular-glue studies.
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- Drug Research
- Biotinylated CRBN/DDB1
- CRL4
- E3 ligase
- PROTAC
- molecular glue
- TR-FRET
- ternary complex
- UA080262
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